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BTRX-335140

BTRX-335140 is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

453.55

Molecular Formula

C25H32FN5O2

Notes

Research use only, not for human use.

Receptor

Δ-opioid receptor|κ-opioid receptor|μ-opioid receptor

CAS Number

2244614-14-8

Available Sizes

Curated Selection

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