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Lerociclib dihydrochloride

Lerociclib dihydrochloride is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 2 nM and 1 nM for CDK6/CyclinD3 and CDK4/CyclinD1, respectively.

Product Specifications

CAS Number

2097938-59-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

547.52

Molecular Formula

C26H36Cl2N8O

Notes

Research use only, not for human use.

Receptor

Cdk4/cyclin D1|cdk6/cyclin D3|CDK9/Cyclin T|CDK5/p35|Cdk5/p25|cdk2/cyclin A|CDK2/cyclinE|CDK1/cyclinB1|CDK7/Cyclin H/MAT1

Available Sizes

Curated Selection

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