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ERK-IN-3

ERK-IN-3 is a potent and orally active inhibitor of ERK. It inhibits ERK1/2 with low single-digit nM IC50 values. It can be used for the research of cancers driven by RAS mutations.

Product Specifications

CAS Number

2055597-12-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

473.93

Molecular Formula

C22H25ClFN7O2

Notes

Research use only, not for human use.

Receptor

ERK1|ERK2

Available Sizes

Curated Selection

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