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PF-543 hydrochloride

PF-543 inhibits SphK1 with a K (i) of 3.6 nM, is sphingosine-competitive and is more than 100-fold selective for SphK1 over the SphK2 isoform.

Product Specifications

CAS Number

1706522-79-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

502.1

Molecular Formula

C27H32ClNO4S

Notes

Research use only, not for human use.

Receptor

SphK1

Available Sizes

Curated Selection

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