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JTE-013

JTE-013 is an effective and specific antagonist of S1P2. JTE-013 suppresses the specific binding of radiolabeled S1P to human and rat S1P2 (IC50s: 17 nM and 22 nM, respectively) .JTE-013 is a S1P2 antagonist. JTE-013 (50-200 μM; 1-3 days) decreased cell viability.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

408.29

Molecular Formula

C17H19Cl2N7O

Notes

Research use only, not for human use.

Receptor

S1P2

CAS Number

383150-41-2

Available Sizes

Curated Selection

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