GSK2807 Trifluoroacetate
GSK2807 Trifluoroacetate is a selective and SAM-competitive inhibitor of SMYD3 (Ki: 14 nM; IC50: 130 nM) .GSK2807, a potent and selective, SAM-competitive inhibitor of SMYD3 (Ki = 14 nM) . A high-resolution crystal structure reveals that GSK2807 bridges the gap between the SAM-binding pocket and the substrate lysine tunnel of SMYD3.
Product Specifications
CAS Number
2245255-66-5
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
566.53
Molecular Formula
C21H33F3N8O7
Notes
Research use only, not for human use.
Receptor
SMYD3
Available Sizes
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items