GSK2807 Trifluoroacetate
GSK2807 Trifluoroacetate is a selective and SAM-competitive inhibitor of SMYD3 (Ki: 14 nM; IC50: 130 nM) .GSK2807, a potent and selective, SAM-competitive inhibitor of SMYD3 (Ki = 14 nM) . A high-resolution crystal structure reveals that GSK2807 bridges the gap between the SAM-binding pocket and the substrate lysine tunnel of SMYD3.
Product Specifications
CAS Number
2245255-66-5
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
566.53
Molecular Formula
C21H33F3N8O7
Notes
Research use only, not for human use.
Receptor
SMYD3
Available Sizes
Curated Selection
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