MK-6892
MK-6892 is a selective and full agonist for the high-affinity nicotinic acid receptor GPR109A (Ki: 4 nM; GTPγS EC50: 16 nM) .MK-6892 evokes a potent internalization of GPR109A in U2OS β-arrestin2-RrGFP cells.MK-6892 shows an EC50 value of 74 nM on calcium mobilization assay.
Product Specifications
CAS Number
917910-45-3
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
386.4
Molecular Formula
C19H22N4O5
Notes
Research use only, not for human use.
Receptor
GPR109A
Available Sizes
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