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MK-6892

MK-6892 is a selective and full agonist for the high-affinity nicotinic acid receptor GPR109A (Ki: 4 nM; GTPγS EC50: 16 nM) .MK-6892 evokes a potent internalization of GPR109A in U2OS β-arrestin2-RrGFP cells.MK-6892 shows an EC50 value of 74 nM on calcium mobilization assay.

Product Specifications

CAS Number

917910-45-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

386.4

Molecular Formula

C19H22N4O5

Notes

Research use only, not for human use.

Receptor

GPR109A

Available Sizes

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