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CTAP (TFA)

CTAP TFA is a potent, highly selective, and brain penetrant antagonist of μ-opioid receptor with IC50 of 3.5 nM. It displays over 1200-fold selectivity over δ opioid (IC50=4500 nM) and somatostatin receptors.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

——

Molecular Formula

——

Notes

Research use only, not for human use.

Receptor

Δ-opioid receptor

Available Sizes

Curated Selection

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