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HGPR91 antagonist 1

HGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM) .GPR91, a 7TM G-Protein-Coupled Receptor, has been recently deorphanized with succinic acid as its endogenous ligand. Current literature indicates that GPR91 plays role in various pathophysiology including renal hypertension, autoimmune disease and retinal angiogenesis.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

529.53

Molecular Formula

C31H23F4N3O

Notes

Research use only, not for human use.

Receptor

HGPR91

CAS Number

1314796-00-3

Available Sizes

Curated Selection

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