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ESI-05

ESI-05 is a specific EPAC2 (exchange protein directly activated by cAMP 2) antagonist (IC50: 0.4 µM) . ESI-05 inhibits cAMP-mediated activation of EPAC2, as well as EAPC2, mediated Rap1 activation.

Product Specifications

CAS Number

5184-64-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

274.38

Molecular Formula

C16H18O2S

Notes

Research use only, not for human use.

Receptor

EPAC2

Available Sizes

Curated Selection

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