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Cabergoline

Cabergoline is an ergot derived-dopamine D2-like receptor agonist. It has high affinity for D2, D3, and 5-HT2B receptors (Ki=0.7, 1.5, and 1.2, respectively) .Cabergoline permits rapid and effective hormonal and tumor control by normalizing prolactin-producing pituitary adenomas levels.Cabergoline acts as a potent agonist of D2, D3 and 5-HT2B receptors.

Product Specifications

CAS Number

81409-90-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

451.60

Molecular Formula

C26H37N5O2

Notes

Research use only, not for human use.

Receptor

D2|D3|5-HT2B

Available Sizes

Frequently Asked Questions

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