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GRP-60367

GRP-60367 is the first small molecule rabies virus (RABV) entry inhibitor, which has nanomolar effect on some RABV strains.Grp-60367 inhibits the entry of a subset of the RABV strain.Grp-60367 showed the specificity and effective anti-RABV activity of the scaffold. In the dose-response analysis, the EC50s range from 2 to 52 nM in different host cell lines.

Product Specifications

CAS Number

1309241-34-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

353.46

Molecular Formula

C21H27N3O2

Notes

Research use only, not for human use.

Receptor

RABV

Available Sizes

Curated Selection

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