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Idelalisib (b)

Idelalisib is a selective inhibitor of p110δ (IC50 : 2.5 nM; in cell-free assays) ; shown to have 40- to 300-fold greater selectivity for p110δ than p110α/β/γ, and 400- to 4000-fold more selectivity to p110δ than C2β, hVPS34, DNA-PK and mTOR.

Product Specifications

CAS Number

1146702-54-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

415.42

Molecular Formula

C22H18FN7O

Notes

Research use only, not for human use.

Receptor

P110δ

Available Sizes

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