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VU591

VU591 is the first reported selective, small-molecule ROMK inhibitor (IC50 of 0.24 μM) . It inhibits potassium transport in isolated perfused rat collecting duct tubules with no effect on sodium transport.

Product Specifications

CAS Number

1222810-74-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

368.3

Molecular Formula

C16H12N6O5

Notes

Research use only, not for human use.

Receptor

Kir1.1|ROMK

Available Sizes

Curated Selection

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