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Taltirelin acetate

Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) (IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release) ) .

Product Specifications

CAS Number

1549593-23-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

465.46

Molecular Formula

C19H27N7O7

Notes

Research use only, not for human use.

Receptor

THR

Available Sizes

Frequently Asked Questions

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