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[Pyr1]-Apelin-13

[Pyr1]-Apelin-13 is a potent and selective endogenous Apelin receptor (APJ) agonist.[Pyr1]-apelin-13 encapsulation in lipoPEG particles (lipoPEG-PA13) results in sustained and extended drug release under physiological conditions[1].[Pyr1]-apelin-13 nanocarriers in a mouse model of pressure-overload induced heart failure demonstrate a sustainable long-term effect of [Pyr1]-apelin-13 in preventing cardiac dysfunction.

Product Specifications

CAS Number

217082-60-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

1533.8

Molecular Formula

C69H108N22O16S

Notes

Research use only, not for human use.

Receptor

Endogenous apelin receptor

Available Sizes

Curated Selection

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