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GW 6471

GW6471 is an antagonist of PPARα with IC50 of 0.24 μ M. GW6471 enhances the binding affinity of the PPAR α ligand-binding domain to the co-repressor proteins SMRT and NCoR.A specific PPARα antagonist.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

619.67

Molecular Formula

C35H36F3N3O4

Notes

Research use only, not for human use.

Receptor

PPARα

CAS Number

880635-03-0

Available Sizes

Curated Selection

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