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MYCi361

MYCi361 is an inhibitor of MYC (binding to MYC with Kd of 3.2 μM) . MYCi361 is a small-molecule MYC inhibitors that inhibits the viability of MYC-dependent cancer cells including prostate cancer (MycCaP, LNCaP, and PC3), leukemia (MV4-11), lymphoma (HL-60 and P493-6), and neuroblastoma (SK-N-B2) with low-micromolar IC50 values.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

594.86

Molecular Formula

C26H16ClF9N2O2

Notes

Research use only, not for human use.

Receptor

MYC

CAS Number

2289690-31-7

Available Sizes

Curated Selection

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