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LDK378 dihydrochloride

Ceritinib dihydrochloride is a selective, orally bioavailable and ATP-competitive inhibitor of ALK tyrosine kinase (IC50 of 200 pM), and also inhibits IGF-1R, InsR, and STK22D (IC50 values of 8, 7, and 23 nM, respectively) .

Product Specifications

CAS Number

1380575-43-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

631.06

Molecular Formula

C28H38Cl3N5O3S

Notes

Research use only, not for human use.

Receptor

ALK

Available Sizes

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