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Taltirelin

Taltirelin is at thyrotropin-releasing hormone receptor (TRH-R) superagonist (IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release) .

Product Specifications

CAS Number

103300-74-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

405.41

Molecular Formula

C17H23N7O5

Notes

Research use only, not for human use.

Receptor

Thyrotropin-releasing hormone receptor

Available Sizes

Frequently Asked Questions

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