Tenalisib (RP6530)
Tenalisib shows selectivity over PI3K α (>300-fold) and β (>100-fold) isoforms. Tenalisib exhibits modest proliferation inhibition in both HEL-RS and HEL-RR cells.
Product Specifications
CAS Number
1639417-53-0
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
415.42
Molecular Formula
C₂₃H₁₈FN₅O₂
Notes
Research use only, not for human use.
Receptor
PI3Kδ, PI3Kγ
Available Sizes
Frequently Asked Questions
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