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Guan-fu base A

Guanfu base A is a potent noncompetitive CYP2D6 inhibitor (Ki: 1.20 μM in HLMs; Ki: 0.37 μM for rCYP2D6) . It also inhibits HERG channel current.

Product Specifications

CAS Number

1394-48-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

429.5

Molecular Formula

C24H31NO6

Notes

Research use only, not for human use.

Receptor

CYP2D6| HERG channel

Available Sizes

Curated Selection

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