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ICA-121431

ICA-121431 is a nanomolar potent small molecule Nav1.7 channel inhibitor with IC50 of 19 nM for rat Nav1.7 with little or no activity against human Nav1.5 or Nav1.7 channels.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

449.55

Molecular Formula

C23H19N3O3S2

Notes

Research use only, not for human use.

Receptor

Nav1.7 channel

CAS Number

313254-51-2

Available Sizes

Curated Selection

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