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ICA-121431

ICA-121431 is a nanomolar potent small molecule Nav1.7 channel inhibitor with IC50 of 19 nM for rat Nav1.7 with little or no activity against human Nav1.5 or Nav1.7 channels.

Product Specifications

CAS Number

313254-51-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

449.55

Molecular Formula

C23H19N3O3S2

Notes

Research use only, not for human use.

Receptor

Nav1.7 channel

Available Sizes

Curated Selection

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