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Gestrinone

Gestrinone is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis. It inhibits leiomyoma cells with an IC50 of 43.67 μM.

Product Specifications

CAS Number

16320-04-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

308.41

Molecular Formula

C21H24O2

Notes

Research use only, not for human use.

Receptor

ER

Available Sizes

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