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TG4-155

TG4-155 is a brain penetrant EP2 antagonist (KB = 2.4 nM) that is over 1000-fold less effective at EP4 (KB = 11.4 µM) and a panel of other receptors and channels.

Product Specifications

CAS Number

1164462-05-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

394.47

Molecular Formula

C23H26N2O4

Notes

Research use only, not for human use.

Receptor

EP2

Available Sizes

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