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Varlitinib

Varlitinib is a selective and potent ErbB1 (EGFR) and ErbB2 (HER2) inhibitor with IC50 of 7 nM and 2 nM respectively. Phase 2.

Product Specifications

CAS Number

845272-21-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

466.94

Molecular Formula

C22H19ClN6O2S

Notes

Research use only, not for human use.

Receptor

EGFR/ErbB1| HER2/ErbB2

Available Sizes

Curated Selection

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