ML221
ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in the β-arrestin assay, and EC80 of 10 nM in both assays.
Product Specifications
CAS Number
877636-42-5
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
385.35
Molecular Formula
C17H11N3O6S
Notes
Research use only, not for human use.
Receptor
APJ
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
CPBT-66021RA 1 mg
Rabbit F(Ab')2 Anti Rat Igg Polyclonal Antibody,FITC
Sign In for Pricing
View Details 
K0803208 1.0 µg DNA
FRA3D sgRNA CRISPR/Cas9 All-in-One Lentivector (Human) (Target 3)
Sign In for Pricing
View Details 45877061 1.0 µg DNA
SUMO2P4 Lentiviral Vector (Human) (CMV) (pLenti-GIII-CMV)
Sign In for Pricing
View Details 
RR208766L3V 200 µL
Gpr151 (NM_181633) Rat Tagged ORF Clone Lentiviral Particle
Sign In for Pricing
View Details