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CTEP

CTEP (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, shows >1000-fold selectivity over other mGlu receptors.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

391.77

Molecular Formula

C19H13ClF3N3O

Notes

Research use only, not for human use.

Receptor

MGluR5

CAS Number

871362-31-1

Available Sizes

Curated Selection

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