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CL-387785

CL-387785 (EKI785; WAY-EKI 785) is an irreversible inhibitor of EGFR (IC50: 370+/-120 pM) ; is able to overcome resistance caused by the T790M mutation on a functional level.

Product Specifications

CAS Number

194423-06-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

381.23

Molecular Formula

C18H13BrN4O

Notes

Research use only, not for human use.

Receptor

EGFR

Available Sizes

Curated Selection

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