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Lomitapide

Lomitapide is a small molecule inhibitor of microsomal triglyceride transfer protein (MTP), an enzyme located in the lumen of the endoplasmic reticulum responsible for absorbing dietary lipids and transferring triglycerides onto apolipoprotein B (apo-B) in the assembly of very-low-density lipoprotein.

Product Specifications

CAS Number

182431-12-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

692.71

Molecular Formula

C39H37F6N3O2

Notes

Research use only, not for human use.

Receptor

MTP

Available Sizes

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