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CPI-360

CPI-360 is a potent, selective, and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.

Product Specifications

CAS Number

1802175-06-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

437.53

Molecular Formula

C25H31N3O4

Notes

Research use only, not for human use.

Receptor

EZH1

Available Sizes

Frequently Asked Questions

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