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RO 46-8443

RO 46-8443 is the first non-peptide endothelin ETB receptor selective antagonist. RO 46-8443 displays up to 2000-fold selectivity for ETB receptors both in terms of binding inhibitory potency and functional inhibition.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

609.69

Molecular Formula

C31H35N3O8S

Notes

Research use only, not for human use.

Receptor

ET-B

CAS Number

175556-12-4

Available Sizes

Curated Selection

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