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Oclacitinib maleate

Oclacitinib is a novel inhibitor of JAK family members with IC50 ranging from 10 to 99 nM and JAK1-dependent cytokines with IC50 ranging from 36 to 249 nM, which did not inhibit a panel of 38 non-JAK kinases.

Product Specifications

CAS Number

1640292-55-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

453.51

Molecular Formula

C15H23N5O2S·C4H4O4

Notes

Research use only, not for human use.

Receptor

JAK1 |JAK2|TYK2 |JAK3

Available Sizes

Curated Selection

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