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FRAX597

FRAX597 is an effective, ATP-competitive inhibitor of group I PAKs, and for PAK1 (IC50=8 nM), PAK2 (IC50=13 nM), and PAK3 (IC50=19 nM) .

Product Specifications

CAS Number

1286739-19-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

558.1

Molecular Formula

C29H28ClN7OS

Notes

Research use only, not for human use.

Receptor

PAK1| PAK2| PAK2| PAK3

Available Sizes

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