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Saclofen

Saclofen is a sulfonic analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7.8 μM) .

Product Specifications

CAS Number

125464-42-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

249.71

Molecular Formula

C9H12ClNO3S

Notes

Research use only, not for human use.

Receptor

GABAB

Available Sizes

Curated Selection

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