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APY29

APY29 is an allosteric modulator of IRE1α; inhibits IRE1α autophosphorylation (IC50 = 280 nM) and activates IRE1α RNase activity.

Product Specifications

CAS Number

1216665-49-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

332.36

Molecular Formula

C17H16N8

Notes

Research use only, not for human use.

Receptor

IRE1α

Available Sizes

Curated Selection

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