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Uprosertib

Uprosertib (GSK2141795) is a selective, ATP-competitive, and orally bioavailable Akt inhibitor with IC50 of 180 nM, 328 nM, and 38 nM for Akt 1, 2 and 3, respectively. Phase 2.

Product Specifications

CAS Number

1047634-65-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

429.25

Molecular Formula

C18H16Cl2F2N4O2

Notes

Research use only, not for human use.

Receptor

Akt1| Akt2| Akt3

Available Sizes

Curated Selection

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