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KDM5A covalent inhibitor N71

KDM5A covalent inhibitor N71 is an irreversible KDM5A inhibitor (IC50=0.22 uM) that covalently interacts with Cys481.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

522.664

Molecular Formula

C28H34N4O4S

Notes

Research use only, not for human use.

Receptor

Histone Demethylase

Available Sizes

Curated Selection

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