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BRD4 inhibitor Compound V

BRD4 inhibitor Compound V is a domain-selective inhibitor of BRD4 with IC50 of 1.8 uM for BRD4 BD1, displays 6- and 16-fold selectivity for BRD4 over BRD2 and BRD3, respectively.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

442.542

Molecular Formula

C26H27FN6

Notes

Research use only, not for human use.

Receptor

Bromodomain

Available Sizes

Frequently Asked Questions

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