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ZXH-3-26

ZXH-3-26 is a novel BRD4 heterobifunctional small-molecule ligand (PROTAC), shows activity exclusively on the BRD4 BD1 (DC50/5h=5 nM) and spares degradation of BRD2 or BRD3 in cellular degradation assays.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

785.273

Molecular Formula

C38H37ClN8O7S

Notes

Research use only, not for human use.

Receptor

PROTAC

Available Sizes

Curated Selection

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