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JNJ-39393406

JNJ-39393406 is a potent, selective positive allosteric α7 nAChR modulator, potentiates a 100 μM choline-induced rise in intracellular calcium mediated by human α7 channels expressed in GH4C1 cells with EC50 of 660 nM.

Product Specifications

CAS Number

953428-73-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

416.389

Molecular Formula

C19H18F2N6O3

Notes

Research use only, not for human use.

Receptor

NAChR

Available Sizes

Curated Selection

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