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Lotamilast

Lotamilast (RVT 501, E6005) is a potent, selective PDE4 inhibitor with IC50 of 2.8 nM, suppresses the production of various cytokines from human lymphocytes and monocytes with IC50 of 0.49-3.1 nM.

Product Specifications

CAS Number

947620-48-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

472.501

Molecular Formula

C26H24N4O5

Notes

Research use only, not for human use.

Receptor

PDE4|PDE-4

Available Sizes

Frequently Asked Questions

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