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RO-5126766

A potent, first-in-class dual Raf/MEK inhibitor with IC50 of 56 nM/160 nM for C-Raf/MEK1.

Product Specifications

CAS Number

946128-88-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

471.4615

Molecular Formula

C21H18FN5O5S

Notes

Research use only, not for human use.

Receptor

MEK1| B-Raf| B-Raf (V600E) | C-Raf

Available Sizes

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