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Pacritinib

Pacritinib (SB1518) is a potent and selective inhibitor of Janus Kinase 2 (JAK2) and Fms-Like Tyrosine Kinase-3 (FLT3) with IC50s of 23 and 22 nM in cell-free assays, respectively. Phase 3.

Product Specifications

CAS Number

937272-79-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

472.58

Molecular Formula

C28H32N4O3

Notes

Research use only, not for human use.

Receptor

FLT3| FLT3 (D835Y) | JAK2| JAK2 (V617F) | Tyk2| JAK3

Available Sizes

Curated Selection

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