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Oprozomib

Oprozomib (ONX-0912; PR-047) is a potent, orally bioavailable proteasome inhibitor that inhibits chymotrypsin-like (CT-L) activity of 20S proteasome β5/LMP7 with IC50 of 36/82 nM.

Product Specifications

CAS Number

935888-69-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

532.6092

Molecular Formula

C25H32N4O7S

Notes

Research use only, not for human use.

Receptor

20Sproteasome

Available Sizes

Curated Selection

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