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GDC-0879

A potent and selective B-Raf kinase inhibitor with IC50 of 0.13 nM against purified B-Raf V600E and a cellular pERK IC50 of 63 nM in the MALME-3M cell line.

Product Specifications

CAS Number

905281-76-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

334.3718

Molecular Formula

C19H18N4O2

Notes

Research use only, not for human use.

Receptor

B-Raf

Available Sizes

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