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KX2-391

KX2-391, the first clinical Src inhibitor (peptidomimetic class) that targets the peptide substrate site of Src, with GI50 of 9-60 nM in cancer cell lines.

Product Specifications

CAS Number

897016-82-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

431.53

Molecular Formula

C26H29N3O3

Notes

Research use only, not for human use.

Receptor

Src (Hep 3B) | Src (Hep G2) | Src (HuH7) | Src (PLC/PRF/5)

Available Sizes

Frequently Asked Questions

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