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GDC-0152

GDC-0152 is a potent antagonist of XIAP-BIR3, ML-IAP-BIR3, cIAP1-BIR3 and cIAP2-BIR3 with Ki of 28 nM, 14 nM, 17 nM and 43 nM, respectively.

Product Specifications

CAS Number

873652-48-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

498.64

Molecular Formula

C25H34N6O3S

Notes

Research use only, not for human use.

Receptor

CIAP1-BIR3| cIAP2-BIR3| MLXBIR3SG| XIAP-BIR2| XIAP-BIR3

Available Sizes

Frequently Asked Questions

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